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Assay Detail

CHEMBL5261127

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Toxicity
Antiproliferative activity against African green monkey COS7 cells assessed as inhibition of cell growth
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Toxicity
Organism Chlorocebus aethiops
Cell Type COS-7
Confidence 1 — Organism
Curated By Autocuration

Target

COS-7 (CHEMBL614564)
Type CELL-LINE
Organism Chlorocebus aethiops

Publication

Structural Analysis of Chemokine Receptor-Ligand Interactions.
Arimont M, Sun SL, Leurs R, Smit M, de Esch IJP, de Graaf C.
J Med Chem (2017) 60 : 4735 -4779
PubMed 28165741 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 5 7.73 8.05

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL5277802 1 8.05
CHEMBL5268017 1 7.96
CHEMBL5272687 1 7.82
CHEMBL5270110 1 7.54
CHEMBL5273480 1 7.30

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL5277802 EC50 = 9.0 nM 8.05
CHEMBL5268017 EC50 = 11.0 nM 7.96
CHEMBL5272687 EC50 = 15.0 nM 7.82
CHEMBL5270110 EC50 = 29.0 nM 7.54
CHEMBL5273480 EC50 = 50.0 nM 7.30