Assay Detail
Binding
CHEMBL5261591
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Binding affinity to HSP90 (unknown origin)
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 5 — Multiple protein complex / RNA |
| Curated By | Autocuration |
Publication
Isoxazole ring as a useful scaffold in a search for new therapeutic agents.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 2 | 7.73 | 8.35 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL252124 | — | — | 1 | 8.35 |
| CHEMBL365617 | — | — | 1 | 7.11 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL252124 | — | Kd | = | 4.5 | nM | 8.35 |
| CHEMBL365617 | — | Kd | = | 78.0 | nM | 7.11 |