Assay Detail
Functional
CHEMBL5261682
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Cytotoxicity against human KMS-26 cells measured after 8 days
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | KMS-26 |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Inhibition of bromodomain-containing protein 9 for the prevention of epigenetically-defined drug resistance.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 5.63 | 5.68 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5270178 | — | — | 1 | 5.68 |
| CHEMBL5282240 | — | — | 1 | 5.58 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5270178 | — | IC50 | = | 2110.0 | nM | 5.68 |
| CHEMBL5282240 | — | IC50 | = | 2610.0 | nM | 5.58 |