Assay Detail
Functional
CHEMBL5261815
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Cytotoxicity against mouse A20 cells measured after 8 days
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Mus musculus |
| Cell Type | A20 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Inhibition of bromodomain-containing protein 9 for the prevention of epigenetically-defined drug resistance.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 5.31 | 5.46 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5282240 | — | — | 1 | 5.46 |
| CHEMBL5270178 | — | — | 1 | 5.16 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5282240 | — | IC50 | = | 3430.0 | nM | 5.46 |
| CHEMBL5270178 | — | IC50 | = | 7000.0 | nM | 5.16 |