Assay Detail
Binding
CHEMBL5262834
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of FABP5 (unknown origin) by fluorescence polarization assay
6
Total Activities
6
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Adipocyte fatty acid binding protein 4 (FABP4) inhibitors. A comprehensive systematic review.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 6 | 5.16 | 5.92 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL82293 | PALMITIC ACID | -1.0 | 1 | 5.92 |
| CHEMBL184795 | — | — | 1 | 5.52 |
| CHEMBL185595 | — | — | 1 | 5.17 |
| CHEMBL363032 | — | — | 1 | 5.04 |
| CHEMBL364141 | — | — | 1 | 4.77 |
| CHEMBL184817 | — | — | 1 | 4.52 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL82293 | PALMITIC ACID | IC50 | = | 1200.0 | nM | 5.92 |
| CHEMBL184795 | — | IC50 | = | 3000.0 | nM | 5.52 |
| CHEMBL185595 | — | IC50 | = | 6700.0 | nM | 5.17 |
| CHEMBL363032 | — | IC50 | = | 9100.0 | nM | 5.04 |
| CHEMBL364141 | — | IC50 | = | 17000.0 | nM | 4.77 |
| CHEMBL184817 | — | IC50 | = | 30000.0 | nM | 4.52 |