Assay Detail
Binding
CHEMBL5262843
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Displacement of BODIPY 500/510 C4 from human FABP3 expressed in Escherichia coli incubated for 30 mins by FP assay
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Adipocyte fatty acid binding protein 4 (FABP4) inhibitors. A comprehensive systematic review.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 4 | 5.92 | 6.10 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4560388 | — | — | 1 | 6.10 |
| CHEMBL247920 | — | — | 1 | 5.92 |
| CHEMBL5282728 | — | — | 1 | 5.89 |
| CHEMBL5282255 | — | — | 1 | 5.77 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4560388 | — | IC50 | = | 800.0 | nM | 6.10 |
| CHEMBL247920 | — | IC50 | = | 1200.0 | nM | 5.92 |
| CHEMBL5282728 | — | IC50 | = | 1300.0 | nM | 5.89 |
| CHEMBL5282255 | — | IC50 | = | 1700.0 | nM | 5.77 |