Assay Detail
Binding
CHEMBL5264185
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of human NTPDase1
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Ectonucleoside triphosphate diphosphohydrolase 1 (CHEMBL5722) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Recent advances in small molecule based cancer immunotherapy.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 6.80 | 7.30 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5277365 | — | — | 1 | 7.30 |
| CHEMBL5283491 | — | — | 1 | 6.30 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5277365 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL5283491 | — | IC50 | = | 500.0 | nM | 6.30 |