Assay Detail
Functional
CHEMBL5317601
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Antiproliferative activity against mouse CT26 cells assessed as inhibition of cell growth measured after 6 days by CellTiter-Glo luminescent assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Mus musculus |
| Cell Type | CT26 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Discovery of the Potent and Highly Selective PARP7 Inhibitor as a Novel Immunotherapeutic Agent for Tumors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 4.96 | 5.20 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5095043 | ATAMPARIB | 1.0 | 1 | 5.20 |
| CHEMBL5395820 | — | — | 1 | 4.71 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5095043 | ATAMPARIB | IC50 | = | 6330.0 | nM | 5.20 |
| CHEMBL5395820 | — | IC50 | = | 19470.0 | nM | 4.71 |