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Assay Detail

CHEMBL5325870

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of glutathione reductase (unknown origin)
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Glutathione reductase, mitochondrial (CHEMBL2755)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Pleiotropic effects of a mitochondrion-targeted glutathione reductase inhibitor on restraining tumor cells.
Zhang R, Xiao N, Xu Q, Gong Q, Kong F, Jiang H.
Eur J Med Chem (2023) 248 : 115069 -115069
PubMed 36610249 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 2 6.23 6.23

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL5425052 1 6.23
CHEMBL5403853 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL5425052 IC50 = 590.0 nM 6.23
CHEMBL5403853 IC50 - -