Assay Detail
Binding
CHEMBL5326170
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of ARFGAP1 (unknown origin)
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
ADP-ribosylation factor GTPase-activating protein 1 (CHEMBL5465332) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Ras superfamily GTPase activating proteins in cancer: Potential therapeutic targets?
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 1 | 6.30 | 6.30 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL259181 | — | — | 1 | 6.30 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL259181 | — | EC50 | = | 500.0 | nM | 6.30 |