Assay Detail
Binding
CHEMBL5331258
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Binding affinity to BCL1 (unknown origin) assessed as inhibition constant by measuring imipenem hydrolysis
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Recent advances in β-lactamase inhibitor chemotypes and inhibition modes.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 4.36 | 4.44 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4639950 | — | — | 1 | 4.44 |
| CHEMBL5267944 | — | — | 1 | 4.28 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4639950 | — | Ki | = | 36000.0 | nM | 4.44 |
| CHEMBL5267944 | — | Ki | = | 53000.0 | nM | 4.28 |