Assay Detail
Binding
CHEMBL5331329
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Binding affinity to Acinetobacter derived cephalosporinase 7 assessed as inhibition constant
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Acinetobacter |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Recent advances in β-lactamase inhibitor chemotypes and inhibition modes.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 3 | 8.13 | 9.35 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3613796 | — | — | 1 | 9.35 |
| CHEMBL257468 | — | — | 1 | 7.68 |
| CHEMBL3586553 | — | — | 1 | 7.35 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3613796 | — | Ki | = | 0.45 | nM | 9.35 |
| CHEMBL257468 | — | Ki | = | 21.0 | nM | 7.68 |
| CHEMBL3586553 | — | Ki | = | 45.0 | nM | 7.35 |