Assay Detail
Binding
CHEMBL5331484
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antagonist activity at 125I-labeled CCK-33 in rat pancreas
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Rattus norvegicus |
| Tissue | Pancreas |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Recent progress toward developing axial chirality bioactive compounds.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 5.85 | 5.85 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL283117 | ASPERLICIN | — | 1 | 5.85 |
| CHEMBL316561 | PROGLUMIDE | 4.0 | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL283117 | ASPERLICIN | IC50 | = | 1400.0 | nM | 5.85 |
| CHEMBL316561 | PROGLUMIDE | IC50 | = | 600000.0 | nM | - |