Assay Detail
Toxicity
CHEMBL5332082
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Cytotoxicity against human GES1 cells assessed as inhibition of cell growth incubated for 72 hrs by SRB assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Toxicity |
| Organism | Homo sapiens |
| Cell Type | GES1 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Discovery of a novel piperlongumine analogue as a microtubule polymerization inhibitor with potent anti-angiogenic and anti-metastatic efficacy.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 5.33 | 5.33 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5419960 | — | — | 1 | 5.33 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5419960 | — | IC50 | = | 4732.0 | nM | 5.33 |