Assay Detail
Binding
CHEMBL5332378
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Binding affinity to beta-Catenin (unknown origin) assessed as dissociation constant by isothermal titration calorimetry
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Recent advances of β-catenin small molecule inhibitors for cancer therapy: Current development and future perspectives.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 2 | 6.37 | 6.38 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3260853 | — | — | 1 | 6.38 |
| CHEMBL254381 | — | — | 1 | 6.35 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3260853 | — | Kd | = | 418.0 | nM | 6.38 |
| CHEMBL254381 | — | Kd | = | 450.0 | nM | 6.35 |