Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL5333647

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of human telomerase incubated for 20 mins by TRAP assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Telomerase reverse transcriptase (CHEMBL2916)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Telomerase: A prominent oncological target for development of chemotherapeutic agents.
Vishwakarma K, Dey R, Bhatt H.
Eur J Med Chem (2023) 249 : 115121 -115121
PubMed 36669398 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 6.94 6.94

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL336434 1 6.94

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL336434 IC50 = 115.0 nM 6.94