Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL5335043

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against DENV-3 H87 infected in african green monkey Vero cells incubated for 24 hrs measured after 3 days post infection
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism dengue virus type 3
Cell Type Vero
Confidence 1 — Organism
Curated By Autocuration

Target

dengue virus type 3 (CHEMBL612717)
Type ORGANISM
Organism dengue virus type 3

Publication

Discovery of Acyl-Indole Derivatives as Pan-Serotype Dengue Virus NS4B Inhibitors.
Kesteleyn B, Bardiot D, Bonfanti JF, De Boeck B, Goethals O, Kaptein SJF, Stoops B, Coesemans E, Fortin J, Muller P, Doublet F, Carlens G, Koukni M, Smets W, Raboisson P, Chaltin P, Simmen K, Van Loock M, Neyts J, Marchand A, Jonckers THM.
J Med Chem (2023) 66 : 8808 -8821
PubMed 37389813 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 4 6.79 7.58

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL5408964 1 7.58
CHEMBL5415953 1 7.20
CHEMBL5400299 1 6.38
CHEMBL4203293 1 6.00

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL5408964 EC50 = 26.0 nM 7.58
CHEMBL5415953 EC50 = 63.0 nM 7.20
CHEMBL5400299 EC50 = 420.0 nM 6.38
CHEMBL4203293 EC50 = 1000.0 nM 6.00