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Assay Detail

CHEMBL5336308

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against SARS-CoV-2 Omicron assessed as reduction of viral growth
8
Total Activities
8
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Severe acute respiratory syndrome coronavirus 2
Confidence 1 — Organism
Curated By Autocuration

Target

SARS-CoV-2 (CHEMBL4303835)
Type ORGANISM
Organism Severe acute respiratory syndrome coronavirus 2

Publication

Bench-to-bedside: Innovation of small molecule anti-SARS-CoV-2 drugs in China.
Yang L, Wang Z.
Eur J Med Chem (2023) 257 : 115503 -115503
PubMed 37229831 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 8 7.50 7.62

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL5404334 1 7.62
CHEMBL4802135 NIRMATRELVIR 4.0 1 7.48
CHEMBL4796938 1 7.48
CHEMBL5174111 1 7.48
CHEMBL5423923 1 7.48
CHEMBL5076204 1 7.48
CHEMBL5267069 1 7.48
CHEMBL5173274 1 7.48

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL5404334 EC50 = 24.0 nM 7.62
CHEMBL4802135 NIRMATRELVIR EC50 = 33.0 nM 7.48
CHEMBL4796938 EC50 = 33.0 nM 7.48
CHEMBL5174111 EC50 = 33.0 nM 7.48
CHEMBL5423923 EC50 = 33.0 nM 7.48
CHEMBL5076204 EC50 = 33.0 nM 7.48
CHEMBL5267069 EC50 = 33.0 nM 7.48
CHEMBL5173274 EC50 = 33.0 nM 7.48