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Assay Detail

CHEMBL5336392

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against SARS-CoV-2 WA1 infected in human A549-hACE2-TMPRSS2 cells assessed as reduction in viral replication
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Severe acute respiratory syndrome coronavirus 2
Confidence 1 — Organism
Curated By Autocuration

Target

SARS-CoV-2 (CHEMBL4303835)
Type ORGANISM
Organism Severe acute respiratory syndrome coronavirus 2

Publication

The research progress of SARS-CoV-2 main protease inhibitors from 2020 to 2022.
Pang X, Xu W, Liu Y, Li H, Chen L.
Eur J Med Chem (2023) 257 : 115491 -115491
PubMed 37244162 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 2 5.68 5.69

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL5173559 1 5.69
CHEMBL5401551 1 5.67

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL5173559 EC50 = 2050.0 nM 5.69
CHEMBL5401551 EC50 = 2150.0 nM 5.67