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Assay Detail

CHEMBL5337740

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of LSD1 (unknown origin)
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Lysine-specific histone demethylase 1A (CHEMBL6136)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Research progress of LSD1-based dual-target agents for cancer therapy.
Yang X.
Bioorg Med Chem (2024) 101 : 117651 -117651
PubMed 38401457 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 7.20 7.20

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL5182796 1 7.20

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL5182796 IC50 = 63.0 nM 7.20