Assay Detail
Binding
CHEMBL5338516
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Inhibition of CREBBP (unknown origin) by TR-FRET assay
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
The Science and Art of Structure-Based Virtual Screening.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 5.91 | 6.52 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3321809 | — | — | 1 | 6.52 |
| CHEMBL5199076 | LUNRESERTIB | 2.0 | 1 | 6.52 |
| CHEMBL3810303 | — | — | 1 | 4.70 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3321809 | — | IC50 | = | 300.0 | nM | 6.52 |
| CHEMBL5199076 | LUNRESERTIB | IC50 | = | 300.0 | nM | 6.52 |
| CHEMBL3810303 | — | IC50 | = | 20000.0 | nM | 4.70 |