Assay Detail
Binding
CHEMBL5342201
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antagonist activity at human TLR2/TLR6
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 7 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Small-Molecule Modulators Targeting Toll-like Receptors for Potential Anticancer Therapeutics.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 5.25 | 5.25 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3935646 | — | — | 1 | 5.25 |
| CHEMBL1313485 | — | — | 1 | 5.24 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3935646 | — | IC50 | = | 5600.0 | nM | 5.25 |
| CHEMBL1313485 | — | IC50 | = | 5700.0 | nM | 5.24 |