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Assay Detail

CHEMBL5348071

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against HCV assessed as reduction in viral growth
6
Total Activities
6
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Hepacivirus hominis
Confidence 1 — Organism
Curated By Autocuration

Target

Hepatitis C virus (CHEMBL379)
Type ORGANISM
Organism Hepacivirus hominis

Publication

Insight into non-nucleoside triazole-based systems as viral polymerases inhibitors.
Bivacqua R, Barreca M, Spanò V, Raimondi MV, Romeo I, Alcaro S, Andrei G, Barraja P, Montalbano A.
Eur J Med Chem (2023) 249 : 115136 -115136
PubMed 36708678 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 6 7.32 7.82

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL230744 1 7.82
CHEMBL509746 1 7.80
CHEMBL490672 FILIBUVIR 3.0 1 7.39
CHEMBL516051 1 7.23
CHEMBL490671 1 7.17
CHEMBL489295 1 6.51

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL230744 EC50 = 15.0 nM 7.82
CHEMBL509746 EC50 = 16.0 nM 7.80
CHEMBL490672 FILIBUVIR EC50 = 41.0 nM 7.39
CHEMBL516051 EC50 = 59.0 nM 7.23
CHEMBL490671 EC50 = 67.0 nM 7.17
CHEMBL489295 EC50 = 310.0 nM 6.51