Assay Detail
Functional
CHEMBL5348352
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Anticancer activity against human G-401 cells assessed as cell growth inhibition
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | G-401 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Triazole-fused pyrimidines in target-based anticancer drug discovery.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 4.78 | 5.48 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4096234 | — | — | 1 | 5.48 |
| CHEMBL4065484 | — | — | 1 | 4.07 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4096234 | — | IC50 | = | 3280.0 | nM | 5.48 |
| CHEMBL4065484 | — | IC50 | = | 85000.0 | nM | 4.07 |