Assay Detail
Functional
CHEMBL5352591
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Antiproliferative activity against human PANC-1 cells assessed as inhibition of cell growth measured after 72 hrs by XTT assay
16
Total Activities
16
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | PANC-1 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Identification of new FK866 analogues with potent anticancer activity against pancreatic cancer.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 16 | 8.79 | 10.10 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5411308 | — | — | 1 | 10.10 |
| CHEMBL5435400 | — | — | 1 | 9.70 |
| CHEMBL5396938 | — | — | 1 | 9.40 |
| CHEMBL566757 | DAPORINAD | 2.0 | 1 | 9.22 |
| CHEMBL5411332 | — | — | 1 | 9.22 |
| CHEMBL5401413 | — | — | 1 | 9.05 |
| CHEMBL5408569 | — | — | 1 | 8.89 |
| CHEMBL5410343 | — | — | 1 | 8.72 |
| CHEMBL5409112 | — | — | 1 | 8.70 |
| CHEMBL5399830 | — | — | 1 | 8.64 |
| CHEMBL5420600 | — | — | 1 | 8.55 |
| CHEMBL5403829 | — | — | 1 | 8.49 |
| CHEMBL5431482 | — | — | 1 | 8.24 |
| CHEMBL5431996 | — | — | 1 | 8.07 |
| CHEMBL5425840 | — | — | 1 | 7.85 |
| CHEMBL5430148 | — | — | 1 | 7.80 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5411308 | — | IC50 | = | 0.08 | nM | 10.10 |
| CHEMBL5435400 | — | IC50 | = | 0.2 | nM | 9.70 |
| CHEMBL5396938 | — | IC50 | = | 0.4 | nM | 9.40 |
| CHEMBL566757 | DAPORINAD | IC50 | = | 0.6 | nM | 9.22 |
| CHEMBL5411332 | — | IC50 | = | 0.6 | nM | 9.22 |
| CHEMBL5401413 | — | IC50 | = | 0.9 | nM | 9.05 |
| CHEMBL5408569 | — | IC50 | = | 1.3 | nM | 8.89 |
| CHEMBL5410343 | — | IC50 | = | 1.9 | nM | 8.72 |
| CHEMBL5409112 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL5399830 | — | IC50 | = | 2.3 | nM | 8.64 |
| CHEMBL5420600 | — | IC50 | = | 2.8 | nM | 8.55 |
| CHEMBL5403829 | — | IC50 | = | 3.2 | nM | 8.49 |
| CHEMBL5431482 | — | IC50 | = | 5.7 | nM | 8.24 |
| CHEMBL5431996 | — | IC50 | = | 8.6 | nM | 8.07 |
| CHEMBL5425840 | — | IC50 | = | 14.0 | nM | 7.85 |
| CHEMBL5430148 | — | IC50 | = | 16.0 | nM | 7.80 |