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Assay Detail

CHEMBL5352879

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiplasmodial activity against Plasmodium falciparum NF54 gametocytes infected in human erythrocyte assessed as inhibition of parasite growthVincubated for 48 hrs by SYBR Green dye based fluorescence assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Plasmodium falciparum
Cell Type Erythrocyte
Confidence 1 — Organism
Curated By Autocuration

Target

Plasmodium falciparum (CHEMBL364)
Type ORGANISM
Organism Plasmodium falciparum

Publication

New structural classes of antimalarials.
Rathod GK, Jain M, Sharma KK, Das S, Basak A, Jain R.
Eur J Med Chem (2022) 242 : 114653 -114653
PubMed 35985254 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 7.71 7.71

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL119096 CRYPTOLEPINE 1 7.71

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL119096 CRYPTOLEPINE IC50 = 19.65 nM 7.71