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Assay Detail

CHEMBL5355402

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of human CGRP1
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Calcitonin gene-related peptide type 1 receptor (CHEMBL3798)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Resveratrol derivatives: Synthesis and their biological activities.
Grau L, Soucek R, Pujol MD.
Eur J Med Chem (2023) 246 : 114962 -114962
PubMed 36463729 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 2 5.59 5.62

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL5431521 1 5.62
CHEMBL5424856 1 5.56

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL5431521 IC50 = 2413.0 nM 5.62
CHEMBL5424856 IC50 = 2772.0 nM 5.56