Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL5355446

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antileishmanial activity against Leishmania panamensis MHOM/CO/87/UA140-EpiR-GFP strain amastigotes assessed as inhibition of parasite growth incubated for 72 hrs by flow cytometric analysis
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Leishmania panamensis
Confidence 1 — Organism
Curated By Autocuration

Target

Leishmania panamensis (CHEMBL612882)
Type ORGANISM
Organism Leishmania panamensis

Publication

Small molecules containing chalcogen elements (S, Se, Te) as new warhead to fight neglected tropical diseases.
Henriquez-Figuereo A, Morán-Serradilla C, Angulo-Elizari E, Sanmartín C, Plano D.
Eur J Med Chem (2023) 246 : 115002 -115002
PubMed 36493616 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 3 5.00 5.17

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL5177826 1 5.17
CHEMBL5409781 1 4.96
CHEMBL5434366 1 4.86

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL5177826 IC50 = 6720.0 nM 5.17
CHEMBL5409781 IC50 = 10920.0 nM 4.96
CHEMBL5434366 IC50 = 13930.0 nM 4.86