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Assay Detail

CHEMBL5357335

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of human DHFR using DHF as substrate assessed as inhibition constant in presence of NADPH by UV-Vis spectrometry analysis
9
Total Activities
9
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Dihydrofolate reductase (CHEMBL202)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Discovery of rigid biphenyl <i>Plasmodium falciparum</i> DHFR inhibitors using a fragment linking strategy.
Hoarau M, Sermmai P, Varatthan T, Thiabma R, Jantra T, Rattanajak R, Vitsupakorn D, Vanichtanankul J, Saepua S, Yuthavong Y, Thongpanchang C, Kamchonwongpaisan S.
RSC Med Chem (2023) 14 : 1755 -1766
PubMed 37731689 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 9 7.18 7.78

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL5421199 1 7.78
CHEMBL3040038 1 7.76
CHEMBL5415214 1 7.71
CHEMBL5432011 1 7.66
CHEMBL5397904 1 6.96
CHEMBL5406769 1 6.86
CHEMBL5417784 1 6.83
CHEMBL5404134 1 6.67
CHEMBL5440218 1 6.37

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL5421199 Ki = 16.58 nM 7.78
CHEMBL3040038 Ki = 17.41 nM 7.76
CHEMBL5415214 Ki = 19.4 nM 7.71
CHEMBL5432011 Ki = 22.0 nM 7.66
CHEMBL5397904 Ki = 108.4 nM 6.96
CHEMBL5406769 Ki = 139.78 nM 6.86
CHEMBL5417784 Ki = 147.13 nM 6.83
CHEMBL5404134 Ki = 214.41 nM 6.67
CHEMBL5440218 Ki = 422.92 nM 6.37