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Assay Detail

CHEMBL5361452

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of Saccharomyces cerevisiae alpha-glucosidase type I using p-nitrophenyl-alpha-D-glucopyranoside as substrate preincubated for 10 mins followed by substrate addition and measured after 30 mins by absorbance based analysis
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Saccharomyces cerevisiae
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

Synthetic α-glucosidase inhibitors as promising anti-diabetic agents: Recent developments and future challenges.
Mushtaq A, Azam U, Mehreen S, Naseer MM.
Eur J Med Chem (2023) 249 : 115119 -115119
PubMed 36680985 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 2 4.57 4.71

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4458405 1 4.71
CHEMBL404271 ACARBOSE 4.0 1 4.42

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4458405 IC50 = 19270.0 nM 4.71
CHEMBL404271 ACARBOSE IC50 = 38250.0 nM 4.42