Assay Detail
Binding
CHEMBL5361471
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Inhibition of alpha-glucosidase (unknown origin) using pNPG as substrate by spectrophotometric analysis
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Synthetic α-glucosidase inhibitors as promising anti-diabetic agents: Recent developments and future challenges.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 6.62 | 8.04 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5411815 | — | — | 1 | 8.04 |
| CHEMBL404271 | ACARBOSE | 4.0 | 1 | 7.44 |
| CHEMBL5402914 | — | — | 1 | 4.38 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5411815 | — | IC50 | = | 9.05 | nM | 8.04 |
| CHEMBL404271 | ACARBOSE | IC50 | = | 36.0 | nM | 7.44 |
| CHEMBL5402914 | — | IC50 | = | 41740.0 | nM | 4.38 |