Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL5361645

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of Rac activation in human MDA-MB-231 cells treated for 24 hrs by Western blot analysis
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Cell Type MDA-MB-231
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

Recent updates on 1,2,3-triazole-containing hybrids with in vivo therapeutic potential against cancers: A mini-review.
Zhao S, Liu J, Lv Z, Zhang G, Xu Z.
Eur J Med Chem (2023) 251 : 115254 -115254
PubMed 36893627 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 6.99 6.99

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL5290216 MBQ-167 1.0 1 6.99

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL5290216 MBQ-167 IC50 = 103.0 nM 6.99