Assay Detail
Binding
CHEMBL5361646
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of CDC42 activation in human MDA-MB-231 cells treated for 24 hrs by Western blot analysis
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | MDA-MB-231 |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Cell division control protein 42 homolog (CHEMBL6088) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Recent updates on 1,2,3-triazole-containing hybrids with in vivo therapeutic potential against cancers: A mini-review.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 7.11 | 7.11 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5290216 | MBQ-167 | 1.0 | 1 | 7.11 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5290216 | MBQ-167 | IC50 | = | 78.0 | nM | 7.11 |