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Assay Detail

CHEMBL5361870

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antimalarial activity against Plasmodium falciparum NF54 infected in human erythrocytes assessed as reduction in parasitemia incubated for 48 hrs by [3H]-hypoxanthine based liquid scintillation counting analysis
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Plasmodium falciparum
Cell Type Erythrocyte
Confidence 1 — Organism
Curated By Autocuration

Target

Plasmodium falciparum (CHEMBL364)
Type ORGANISM
Organism Plasmodium falciparum

Publication

Current development of β-carboline derived potential antimalarial scaffolds.
Kushwaha P, Kumar V, Saha B.
Eur J Med Chem (2023) 252 : 115247 -115247
PubMed 36931118 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 9.30 9.30

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1082723 CIPARGAMIN 2.0 1 9.30

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1082723 CIPARGAMIN IC50 = 0.5 nM 9.30