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Assay Detail

CHEMBL5363516

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Cytotoxicity against human MDA-MB-231 cells assessed as reduction in cell viability by CCK-8 assay
6
Total Activities
6
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type MDA-MB-231
Confidence 1 — Organism
Curated By Autocuration

Target

MDA-MB-231 (CHEMBL400)
Type CELL-LINE
Organism Homo sapiens

Publication

Phyllospongianes A-E, Dinorscalarane Sesterterpenes from the Marine Sponge <i>Phyllospongia foliascens</i>.
Yu HB, Hu B, Wu GF, Ning Z, He Y, Jiao BH, Liu XY, Lin HW.
J Nat Prod (2023) 86 : 1754 -1760
PubMed 37335557 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 6 4.74 4.88

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL5399306 1 4.88
CHEMBL810 TEMOZOLOMIDE 4.0 1 4.84
CHEMBL5411947 1 4.49
CHEMBL5437546 1 -
CHEMBL5434354 1 -
CHEMBL5414208 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL5399306 IC50 = 13200.0 nM 4.88
CHEMBL810 TEMOZOLOMIDE IC50 = 14400.0 nM 4.84
CHEMBL5411947 IC50 = 32300.0 nM 4.49
CHEMBL5437546 IC50 > 50000.0 nM -
CHEMBL5434354 IC50 > 50000.0 nM -
CHEMBL5414208 IC50 > 50000.0 nM -