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Assay Detail

CHEMBL5364876

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Functional
Antiproliferative activity against human MV4-11 cells
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type MV4-11
Confidence 1 — Organism
Curated By Autocuration

Target

MV4-11 (CHEMBL613835)
Type CELL-LINE
Organism Homo sapiens

Publication

Drug Discovery Targeting Nuclear Receptor Binding SET Domain Protein 2 (NSD2).
Ma Z, Bolinger AA, Chen H, Zhou J.
J Med Chem (2023) 66 : 10991 -11026
PubMed 37578463 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 5.65 5.65

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL5186268 1 5.65

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL5186268 IC50 = 2230.0 nM 5.65