Assay Detail
Functional
CHEMBL5364877
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antiproliferative activity against human KMS-11 cells assessed as inhibition of cell growth
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | KMS-11 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Drug Discovery Targeting Nuclear Receptor Binding SET Domain Protein 2 (NSD2).
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 5.07 | 5.07 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5186268 | — | — | 1 | 5.07 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5186268 | — | IC50 | = | 8430.0 | nM | 5.07 |