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Assay Detail

CHEMBL5366823

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiproliferative activity against mouse B16 cells assessed as reduction in cell viability incubated for 48 hrs irradiated with 365 nm uv light for 4 min by CCK-8 assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Mus musculus
Cell Type B16
Confidence 1 — Organism
Curated By Autocuration

Target

B16 (CHEMBL381)
Type CELL-LINE
Organism Mus musculus

Publication

Discovery of a photosensitizing PI3K inhibitor for tumor therapy: Design, synthesis and in vitro biological evaluation.
Yang C, Gong Y, Deng M, Ling Y, Wang J, Zhou Y.
Bioorg Med Chem Lett (2023) 94 : 129459 -129459
PubMed 37634762 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 5.06 5.06

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL5438780 1 5.06

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL5438780 IC50 = 8800.0 nM 5.06