Assay Detail
Binding
CHEMBL5368327
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Binding affinity to LXR alpha (unknown origin) by Lanthascreen TR-FRET assay
12
Total Activities
12
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
GNE-235: A Lead Compound Selective for the Second Bromodomain of PBRM1.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 12 | 5.12 | 5.17 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5406315 | — | — | 1 | 5.17 |
| CHEMBL5411199 | — | — | 1 | 5.07 |
| CHEMBL5428009 | — | — | 1 | - |
| CHEMBL5424811 | — | — | 1 | - |
| CHEMBL5177096 | — | — | 1 | - |
| CHEMBL5415064 | — | — | 1 | - |
| CHEMBL5401472 | — | — | 1 | - |
| CHEMBL5425250 | — | — | 1 | - |
| CHEMBL5431862 | — | — | 1 | - |
| CHEMBL5426305 | — | — | 1 | - |
| CHEMBL3752911 | — | — | 1 | - |
| CHEMBL5207330 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5406315 | — | EC50 | = | 6700.0 | nM | 5.17 |
| CHEMBL5411199 | — | EC50 | = | 8600.0 | nM | 5.07 |
| CHEMBL5428009 | — | EC50 | > | 20000.0 | nM | - |
| CHEMBL5424811 | — | EC50 | > | 20000.0 | nM | - |
| CHEMBL5177096 | — | EC50 | > | 20000.0 | nM | - |
| CHEMBL5415064 | — | EC50 | > | 20000.0 | nM | - |
| CHEMBL5401472 | — | EC50 | > | 20000.0 | nM | - |
| CHEMBL5425250 | — | EC50 | > | 20000.0 | nM | - |
| CHEMBL5431862 | — | EC50 | > | 20000.0 | nM | - |
| CHEMBL5426305 | — | EC50 | > | 20000.0 | nM | - |
| CHEMBL3752911 | — | EC50 | > | 20000.0 | nM | - |
| CHEMBL5207330 | — | EC50 | > | 20000.0 | nM | - |