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Assay Detail

CHEMBL5371702

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of G9a (unknown origin)
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Histone-lysine N-methyltransferase EHMT2 (CHEMBL6032)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

NSD3: Advances in cancer therapeutic potential and inhibitors research.
Xiu S, Chi X, Jia Z, Shi C, Zhang X, Li Q, Gao T, Zhang L, Liu Z.
Eur J Med Chem (2023) 256 : 115440 -115440
PubMed 37182335 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 5.72 5.72

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1895209 1 5.72

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1895209 IC50 = 1900.0 nM 5.72