Assay Detail
Binding
CHEMBL5372969
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Displacement of [3H]propionyl-pNPY from human Y2R expressed in CHO cells
24
Total Activities
12
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | CHO |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
[<sup>3</sup>H]UR-JG102-A Radiolabeled Cyclic Peptide with High Affinity and Excellent Selectivity for the Neuropeptide Y Y<sub>4</sub> Receptor.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 24 | 6.04 | 6.04 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5421880 | — | — | 2 | 6.04 |
| CHEMBL5429140 | — | — | 2 | - |
| CHEMBL5422869 | — | — | 2 | - |
| CHEMBL5437701 | — | — | 2 | - |
| CHEMBL5435492 | — | — | 2 | - |
| CHEMBL5400627 | — | — | 2 | - |
| CHEMBL5396128 | — | — | 2 | - |
| CHEMBL5430318 | — | — | 2 | - |
| CHEMBL5398948 | — | — | 2 | - |
| CHEMBL5437695 | — | — | 2 | - |
| CHEMBL5428340 | — | — | 2 | - |
| CHEMBL5423253 | — | — | 2 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5421880 | — | Ki | = | 912.01 | nM | 6.04 |
| CHEMBL5396128 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL5429140 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL5422869 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL5422869 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL5437701 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL5437701 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL5435492 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL5435492 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL5400627 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL5400627 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL5421880 | — | Ki | > | 948.0 | nM | - |
| CHEMBL5429140 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL5430318 | — | Ki | > | 3162.28 | nM | - |
| CHEMBL5430318 | — | Ki | > | 3000.0 | nM | - |
| CHEMBL5398948 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL5398948 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL5437695 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL5437695 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL5428340 | — | Ki | > | 3162.28 | nM | - |
| CHEMBL5428340 | — | Ki | > | 3000.0 | nM | - |
| CHEMBL5423253 | — | Ki | > | 3162.28 | nM | - |
| CHEMBL5423253 | — | Ki | > | 3000.0 | nM | - |
| CHEMBL5396128 | — | Ki | > | 10000.0 | nM | - |