Assay Detail
Functional
CHEMBL5374608
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Cytotoxicity against 12 hrs BODIPY-TZ treated human MCF7 cells assessed as inhbition of cell growth measured after 48 hrs by CCK-8 method
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | MCF7 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Rational Design of Bioorthogonally Activatable PROTAC for Tumor-Targeted Protein Degradation.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 6.58 | 6.58 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5394958 | — | — | 1 | 6.58 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5394958 | — | IC50 | = | 263.6 | nM | 6.58 |