Assay Detail
Functional
CHEMBL5380437
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antiviral activity against Human rhinovirus 14 infected in human H1-HeLa cells incubated for 3 days measured by crystal violet staining based plaque counting analysis
34
Total Activities
34
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | rhinovirus B14 |
| Cell Type | H1-HeLa |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Highly potent and selective phosphatidylinositol 4-kinase IIIβ inhibitors as broad-spectrum anti-rhinoviral agents.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 34 | 6.91 | 8.10 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5403406 | — | — | 1 | 8.10 |
| CHEMBL5435139 | — | — | 1 | 8.00 |
| CHEMBL5431632 | — | — | 1 | 7.80 |
| CHEMBL5402886 | — | — | 1 | 7.70 |
| CHEMBL5432195 | — | — | 1 | 7.66 |
| CHEMBL5431408 | — | — | 1 | 7.55 |
| CHEMBL5439775 | — | — | 1 | 7.55 |
| CHEMBL5427380 | — | — | 1 | 7.50 |
| CHEMBL5395492 | — | — | 1 | 7.47 |
| CHEMBL5410515 | — | — | 1 | 7.46 |
| CHEMBL5431413 | — | — | 1 | 7.41 |
| CHEMBL5435605 | — | — | 1 | 7.39 |
| CHEMBL5428790 | — | — | 1 | 7.33 |
| CHEMBL5426813 | — | — | 1 | 7.28 |
| CHEMBL20210 | RUPINTRIVIR | 2.0 | 1 | 7.24 |
| CHEMBL5437936 | — | — | 1 | 7.17 |
| CHEMBL5425138 | — | — | 1 | 7.16 |
| CHEMBL5423836 | — | — | 1 | 7.14 |
| CHEMBL5415642 | — | — | 1 | 7.11 |
| CHEMBL5428664 | — | — | 1 | 7.10 |
| CHEMBL5411938 | — | — | 1 | 7.06 |
| CHEMBL29609 | PLECONARIL | 2.0 | 1 | 6.55 |
| CHEMBL5396829 | — | — | 1 | 6.50 |
| CHEMBL283403 | ENVIROXIME | 2.0 | 1 | 6.48 |
| CHEMBL1229535 | — | — | 1 | 6.11 |
| CHEMBL5431694 | — | — | 1 | 6.00 |
| CHEMBL5417357 | — | — | 1 | 5.89 |
| CHEMBL5401240 | — | — | 1 | 5.89 |
| CHEMBL5406053 | — | — | 1 | 5.85 |
| CHEMBL5421194 | — | — | 1 | 5.42 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5403406 | — | EC50 | = | 8.0 | nM | 8.10 |
| CHEMBL5435139 | — | EC50 | = | 10.0 | nM | 8.00 |
| CHEMBL5431632 | — | EC50 | = | 16.0 | nM | 7.80 |
| CHEMBL5402886 | — | EC50 | = | 20.0 | nM | 7.70 |
| CHEMBL5432195 | — | EC50 | = | 22.0 | nM | 7.66 |
| CHEMBL5431408 | — | EC50 | = | 28.0 | nM | 7.55 |
| CHEMBL5439775 | — | EC50 | = | 28.0 | nM | 7.55 |
| CHEMBL5427380 | — | EC50 | = | 32.0 | nM | 7.50 |
| CHEMBL5395492 | — | EC50 | = | 34.0 | nM | 7.47 |
| CHEMBL5410515 | — | EC50 | = | 35.0 | nM | 7.46 |
| CHEMBL5431413 | — | EC50 | = | 39.0 | nM | 7.41 |
| CHEMBL5435605 | — | EC50 | = | 41.0 | nM | 7.39 |
| CHEMBL5428790 | — | EC50 | = | 47.0 | nM | 7.33 |
| CHEMBL5426813 | — | EC50 | = | 52.0 | nM | 7.28 |
| CHEMBL20210 | RUPINTRIVIR | EC50 | = | 58.0 | nM | 7.24 |
| CHEMBL5437936 | — | EC50 | = | 67.0 | nM | 7.17 |
| CHEMBL5425138 | — | EC50 | = | 69.0 | nM | 7.16 |
| CHEMBL5423836 | — | EC50 | = | 73.0 | nM | 7.14 |
| CHEMBL5415642 | — | EC50 | = | 78.0 | nM | 7.11 |
| CHEMBL5428664 | — | EC50 | = | 80.0 | nM | 7.10 |
| CHEMBL5411938 | — | EC50 | = | 88.0 | nM | 7.06 |
| CHEMBL29609 | PLECONARIL | EC50 | = | 280.0 | nM | 6.55 |
| CHEMBL5396829 | — | EC50 | = | 320.0 | nM | 6.50 |
| CHEMBL283403 | ENVIROXIME | EC50 | = | 330.0 | nM | 6.48 |
| CHEMBL1229535 | — | EC50 | = | 770.0 | nM | 6.11 |
| CHEMBL5431694 | — | EC50 | = | 1000.0 | nM | 6.00 |
| CHEMBL5417357 | — | EC50 | = | 1300.0 | nM | 5.89 |
| CHEMBL5401240 | — | EC50 | = | 1300.0 | nM | 5.89 |
| CHEMBL5406053 | — | EC50 | = | 1400.0 | nM | 5.85 |
| CHEMBL5421194 | — | EC50 | = | 3800.0 | nM | 5.42 |
| CHEMBL5402263 | — | EC50 | = | 4400.0 | nM | 5.36 |
| CHEMBL5437791 | — | EC50 | = | 14500.0 | nM | 4.84 |
| CHEMBL5401566 | — | EC50 | > | 28.0 | nM | - |
| CHEMBL5402317 | — | EC50 | > | 3700.0 | nM | - |