Assay Detail
Functional
CHEMBL5380438
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antiviral activity against Human rhinovirus 16 infected in human H1-HeLa cells incubated for 3 days measured by crystal violet staining based plaque counting analysis
34
Total Activities
34
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | rhinovirus A16 |
| Cell Type | H1-HeLa |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Highly potent and selective phosphatidylinositol 4-kinase IIIβ inhibitors as broad-spectrum anti-rhinoviral agents.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 34 | 6.79 | 8.15 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5403406 | — | — | 1 | 8.15 |
| CHEMBL5435139 | — | — | 1 | 7.68 |
| CHEMBL5431632 | — | — | 1 | 7.58 |
| CHEMBL5402886 | — | — | 1 | 7.52 |
| CHEMBL5432195 | — | — | 1 | 7.50 |
| CHEMBL5431408 | — | — | 1 | 7.33 |
| CHEMBL5439775 | — | — | 1 | 7.21 |
| CHEMBL5395492 | — | — | 1 | 7.17 |
| CHEMBL5410515 | — | — | 1 | 7.17 |
| CHEMBL5427380 | — | — | 1 | 7.14 |
| CHEMBL5428790 | — | — | 1 | 7.14 |
| CHEMBL5435605 | — | — | 1 | 7.12 |
| CHEMBL5431413 | — | — | 1 | 7.12 |
| CHEMBL20210 | RUPINTRIVIR | 2.0 | 1 | 7.10 |
| CHEMBL5426813 | — | — | 1 | 7.10 |
| CHEMBL5423836 | — | — | 1 | 7.07 |
| CHEMBL5437936 | — | — | 1 | 7.04 |
| CHEMBL5425138 | — | — | 1 | 7.04 |
| CHEMBL5415642 | — | — | 1 | 6.92 |
| CHEMBL5428664 | — | — | 1 | 6.85 |
| CHEMBL29609 | PLECONARIL | 2.0 | 1 | 6.57 |
| CHEMBL283403 | ENVIROXIME | 2.0 | 1 | 6.41 |
| CHEMBL5411938 | — | — | 1 | 6.27 |
| CHEMBL5431694 | — | — | 1 | 6.25 |
| CHEMBL5401240 | — | — | 1 | 6.10 |
| CHEMBL1229535 | — | — | 1 | 6.08 |
| CHEMBL5417357 | — | — | 1 | 6.00 |
| CHEMBL5406053 | — | — | 1 | 5.89 |
| CHEMBL5421194 | — | — | 1 | 5.70 |
| CHEMBL5402263 | — | — | 1 | 5.48 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5403406 | — | EC50 | = | 7.0 | nM | 8.15 |
| CHEMBL5435139 | — | EC50 | = | 21.0 | nM | 7.68 |
| CHEMBL5431632 | — | EC50 | = | 26.0 | nM | 7.58 |
| CHEMBL5402886 | — | EC50 | = | 30.0 | nM | 7.52 |
| CHEMBL5432195 | — | EC50 | = | 32.0 | nM | 7.50 |
| CHEMBL5431408 | — | EC50 | = | 47.0 | nM | 7.33 |
| CHEMBL5439775 | — | EC50 | = | 62.0 | nM | 7.21 |
| CHEMBL5395492 | — | EC50 | = | 67.0 | nM | 7.17 |
| CHEMBL5410515 | — | EC50 | = | 68.0 | nM | 7.17 |
| CHEMBL5427380 | — | EC50 | = | 72.0 | nM | 7.14 |
| CHEMBL5428790 | — | EC50 | = | 73.0 | nM | 7.14 |
| CHEMBL5435605 | — | EC50 | = | 75.0 | nM | 7.12 |
| CHEMBL5431413 | — | EC50 | = | 76.0 | nM | 7.12 |
| CHEMBL20210 | RUPINTRIVIR | EC50 | = | 80.0 | nM | 7.10 |
| CHEMBL5426813 | — | EC50 | = | 80.0 | nM | 7.10 |
| CHEMBL5423836 | — | EC50 | = | 85.0 | nM | 7.07 |
| CHEMBL5425138 | — | EC50 | = | 92.0 | nM | 7.04 |
| CHEMBL5437936 | — | EC50 | = | 91.0 | nM | 7.04 |
| CHEMBL5415642 | — | EC50 | = | 120.0 | nM | 6.92 |
| CHEMBL5428664 | — | EC50 | = | 140.0 | nM | 6.85 |
| CHEMBL29609 | PLECONARIL | EC50 | = | 270.0 | nM | 6.57 |
| CHEMBL283403 | ENVIROXIME | EC50 | = | 390.0 | nM | 6.41 |
| CHEMBL5411938 | — | EC50 | = | 539.0 | nM | 6.27 |
| CHEMBL5431694 | — | EC50 | = | 560.0 | nM | 6.25 |
| CHEMBL5401240 | — | EC50 | = | 790.0 | nM | 6.10 |
| CHEMBL1229535 | — | EC50 | = | 840.0 | nM | 6.08 |
| CHEMBL5417357 | — | EC50 | = | 1000.0 | nM | 6.00 |
| CHEMBL5406053 | — | EC50 | = | 1300.0 | nM | 5.89 |
| CHEMBL5421194 | — | EC50 | = | 2000.0 | nM | 5.70 |
| CHEMBL5402263 | — | EC50 | = | 3300.0 | nM | 5.48 |
| CHEMBL5437791 | — | EC50 | = | 12000.0 | nM | 4.92 |
| CHEMBL5401566 | — | EC50 | > | 28.0 | nM | - |
| CHEMBL5402317 | — | EC50 | > | 3700.0 | nM | - |
| CHEMBL5396829 | — | EC50 | < | 250.0 | nM | - |