Assay Detail
Functional
CHEMBL5381509
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Cytotoxicity against human MV4-11 cells assessed as reduction in cell viability incubated for 24 hrs by celltiter-glo assay
44
Total Activities
44
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | MV4-11 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Optimized M24B Aminopeptidase Inhibitors for CARD8 Inflammasome Activation.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 44 | 5.34 | 6.57 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5410658 | — | — | 1 | 6.57 |
| CHEMBL5438224 | — | — | 1 | 6.37 |
| CHEMBL5399924 | — | — | 1 | 6.35 |
| CHEMBL5401781 | — | — | 1 | 6.22 |
| CHEMBL5397935 | — | — | 1 | 6.19 |
| CHEMBL5419034 | — | — | 1 | 6.18 |
| CHEMBL5400780 | — | — | 1 | 6.08 |
| CHEMBL5436435 | — | — | 1 | 6.00 |
| CHEMBL5402862 | — | — | 1 | 5.89 |
| CHEMBL5437413 | — | — | 1 | 5.66 |
| CHEMBL5393876 | — | — | 1 | 5.52 |
| CHEMBL457092 | BESTATIN METHYL ESTER | — | 1 | 5.41 |
| CHEMBL5415378 | — | — | 1 | 5.27 |
| CHEMBL5433606 | — | — | 1 | 5.25 |
| CHEMBL5419938 | — | — | 1 | 5.14 |
| CHEMBL5430934 | — | — | 1 | 5.09 |
| CHEMBL5403940 | — | — | 1 | 5.09 |
| CHEMBL5404330 | — | — | 1 | 5.00 |
| CHEMBL5429139 | — | — | 1 | 4.96 |
| CHEMBL5398054 | — | — | 1 | 4.85 |
| CHEMBL5406619 | — | — | 1 | 4.82 |
| CHEMBL5433567 | — | — | 1 | 4.82 |
| CHEMBL5419166 | — | — | 1 | 4.77 |
| CHEMBL5415840 | — | — | 1 | 4.72 |
| CHEMBL5435178 | — | — | 1 | 4.46 |
| CHEMBL5394915 | — | — | 1 | 4.34 |
| CHEMBL5421036 | — | — | 1 | 4.22 |
| CHEMBL5407130 | — | — | 1 | 4.21 |
| CHEMBL311875 | — | — | 1 | - |
| CHEMBL5433668 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5410658 | — | IC50 | = | 270.0 | nM | 6.57 |
| CHEMBL5438224 | — | IC50 | = | 430.0 | nM | 6.37 |
| CHEMBL5399924 | — | IC50 | = | 450.0 | nM | 6.35 |
| CHEMBL5401781 | — | IC50 | = | 600.0 | nM | 6.22 |
| CHEMBL5397935 | — | IC50 | = | 650.0 | nM | 6.19 |
| CHEMBL5419034 | — | IC50 | = | 660.0 | nM | 6.18 |
| CHEMBL5400780 | — | IC50 | = | 840.0 | nM | 6.08 |
| CHEMBL5436435 | — | IC50 | = | 1000.0 | nM | 6.00 |
| CHEMBL5402862 | — | IC50 | = | 1300.0 | nM | 5.89 |
| CHEMBL5437413 | — | IC50 | = | 2200.0 | nM | 5.66 |
| CHEMBL5393876 | — | IC50 | = | 3000.0 | nM | 5.52 |
| CHEMBL457092 | BESTATIN METHYL ESTER | IC50 | = | 3900.0 | nM | 5.41 |
| CHEMBL5415378 | — | IC50 | = | 5400.0 | nM | 5.27 |
| CHEMBL5433606 | — | IC50 | = | 5600.0 | nM | 5.25 |
| CHEMBL5419938 | — | IC50 | = | 7300.0 | nM | 5.14 |
| CHEMBL5430934 | — | IC50 | = | 8200.0 | nM | 5.09 |
| CHEMBL5403940 | — | IC50 | = | 8100.0 | nM | 5.09 |
| CHEMBL5404330 | — | IC50 | = | 10000.0 | nM | 5.00 |
| CHEMBL5429139 | — | IC50 | = | 11000.0 | nM | 4.96 |
| CHEMBL5398054 | — | IC50 | = | 14000.0 | nM | 4.85 |
| CHEMBL5406619 | — | IC50 | = | 15000.0 | nM | 4.82 |
| CHEMBL5433567 | — | IC50 | = | 15000.0 | nM | 4.82 |
| CHEMBL5419166 | — | IC50 | = | 17000.0 | nM | 4.77 |
| CHEMBL5415840 | — | IC50 | = | 19000.0 | nM | 4.72 |
| CHEMBL5435178 | — | IC50 | = | 35000.0 | nM | 4.46 |
| CHEMBL5394915 | — | IC50 | = | 46000.0 | nM | 4.34 |
| CHEMBL5421036 | — | IC50 | = | 60000.0 | nM | 4.22 |
| CHEMBL5407130 | — | IC50 | = | 61000.0 | nM | 4.21 |
| CHEMBL5412812 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL5396150 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL5403929 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL5421582 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL5412099 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL5396773 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL5432938 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL5403523 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL5409645 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL5419889 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL5403681 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL5438777 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL5435351 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL5427035 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL5433668 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL311875 | — | IC50 | > | 20000.0 | nM | - |