Assay Detail
Binding
CHEMBL5385490
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Agonist activity at NOR1 (unknown origin) by Gal4 hybrid reporter gene assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Nuclear receptor subfamily 4 group A member 3 (CHEMBL1961792) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Development of a Potent Nurr1 Agonist Tool for In Vivo Applications.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 1 | 5.54 | 5.54 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL197194 | VIDOFLUDIMUS | 3.0 | 1 | 5.54 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL197194 | VIDOFLUDIMUS | EC50 | = | 2900.0 | nM | 5.54 |