Assay Detail
Binding
CHEMBL5385503
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Binding affinity to Nurr1-LBD (unknown origin) by Isothermal titration colorimetry
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Nuclear receptor subfamily 4 group A member 2 (CHEMBL5002) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Development of a Potent Nurr1 Agonist Tool for In Vivo Applications.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 2 | 6.34 | 6.52 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5417085 | — | — | 1 | 6.52 |
| CHEMBL197194 | VIDOFLUDIMUS | 3.0 | 1 | 6.16 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5417085 | — | Kd | = | 300.0 | nM | 6.52 |
| CHEMBL197194 | VIDOFLUDIMUS | Kd | = | 700.0 | nM | 6.16 |