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Assay Detail

CHEMBL5386549

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiproliferative activity against human U373 cells assessed as inhibition of cell growth measured after 72 hrs by CTG assay
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type U373
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

Natural quinazolinones: From a treasure house to promising anticancer leads.
Li H, Fu G, Zhong W.
Eur J Med Chem (2023) 245 : 114915 -114915
PubMed 36375335 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 5 4.05 4.05

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL557488 FUMITREMORGIN F 1 4.05
CHEMBL5436778 1 -
CHEMBL5437139 1 -
CHEMBL5417203 1 -
CHEMBL5437191 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL557488 FUMITREMORGIN F IC50 = 90000.0 nM 4.05
CHEMBL5436778 IC50 > 100000.0 nM -
CHEMBL5437139 IC50 > 100000.0 nM -
CHEMBL5417203 IC50 > 100000.0 nM -
CHEMBL5437191 IC50 > 100000.0 nM -