Assay Detail
Functional
CHEMBL5464241
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Full-length RXR reporter gene assay (RXR RXR Homodimer) (transiently transfected HEK293T cells using firefly lucifease reporter constructs)
1
Total Activities
1
Compounds Tested
1
Activity Types
2
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | HEK293 |
| Confidence | 5 — Multiple protein complex / RNA |
| Curated By | Autocuration |
Publication
Data for DCP probe JP3000
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 1 | 8.59 | 8.59 |
Assay Parameters
| Parameter | Type | Value | Units | Text |
|---|---|---|---|---|
| Additional information | Additional information | - | — | transiently transfected HEK293T cells using firefly lucifease reporter constructs |
| Target protein length | Target protein length | - | — | full length |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5404648 | — | — | 1 | 8.59 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5404648 | — | EC50 | = | 2.6 | nM | 8.59 |