Assay Detail
Binding
CHEMBL5464403
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Inhibition of Vasopressin V1A at 10.0 µM in the Eurofins-Panlabs selectivity screen
3
Total Activities
3
Compounds Tested
2
Activity Types
3
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Data for DCP probe BAY-9835
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 9.30 | 9.30 |
| Inhibition | 1 | - | - |
Assay Parameters
| Parameter | Type | Value | Units | Text |
|---|---|---|---|---|
| Assay publication | Assay publication | - | — | https://www.eurofinsdiscovery.com/catalog/287530 |
| Target protein length | Target protein length | - | — | full length |
| Target protein type | Target protein type | - | — | recombinant |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4594444 | PECAVAPTAN | 2.0 | 1 | 9.30 |
| CHEMBL5465173 | — | — | 1 | - |
| CHEMBL5575976 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4594444 | PECAVAPTAN | Ki | = | 0.5 | nM | 9.30 |
| CHEMBL5465173 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL5575976 | — | Inhibition | = | 7.0 | % | - |